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Synthesis and investigation of FITC-labeled and crizotinib-conjugated GnRH analogues and their relevance in targeted cancer therapy

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Academic year: 2022

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Figure 1.: Structure of FITC-GnRH conjugates.
Table I.: The results of the FITC-GnRH treated cell lines.
Figure 2.: The selected crizotinib analogues for GnRH conjugation.
Figure 3.: pH-dependent membrane permeability of crizotinib, MJ37, MJ55 and  caffeine, measured by PAMPA
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